Kinase
Classification
Activity Assays
Binding Assay
Z'-LYTE®
Adapta®
LanthaScreen®
ABL1
Tyr-C
x
ABL1 E255K
Tyr-C
x
ABL1 G250E
Tyr-C
x
ABL1 T315I
Tyr-C
x
ABL1 Y253F
Tyr-C
x
ABL2 (Arg )
Tyr-C
x
ACVR1 (ALK2 )
Ser/Thr
x
ACVR1B (ALK4 )
Ser/Thr
x
ACVR2B
Ser/Thr
x
ADRBK1 (GRK2 )
Ser/Thr
x
ADRBK2 (GRK3 )
Ser/Thr
x
AKT1 (PKB alpha )
Ser/Thr
x
AKT2 (PKB beta )
Ser/Thr
x
AKT3 (PKB gamma )
Ser/Thr
x
AMPK A1/B1/G1
Ser/Thr
x
AMPK A2/B1/G1
Ser/Thr
x
AURKA (Aurora A )
Ser/Thr
x
AURKB (Aurora B )
Ser/Thr
x
AURKC (Aurora C )
Ser/Thr
x
AXL
Tyr-R
x
BLK
Tyr-C
x
BMPR1A (ALK3 )
Ser/Thr
x
BMX
Tyr-C
x
BRAF
Ser/Thr
x
x
BRAF V599E
Ser/Thr
x
x
BRSK1 (SAD1 )
Ser/Thr
x
BTK
Tyr-C
x
CAMK1 (CaMK1 )
Ser/Thr
x
CAMK1D (CaMKI delta )
Ser/Thr
x
CAMK2A (CaMKII alpha )
Ser/Thr
x
CAMK2B (CaMKII beta )
Ser/Thr
x
CAMK2D (CaMKII delta )
Ser/Thr
x
CAMK4 (CaMKIV )
Ser/Thr
x
CAMKK1 (CAMKKA )
Ser/Thr
x
CAMKK2 (CaMKK beta )
Ser/Thr
x
CDC42 BPA (MRCKA )
Ser/Thr
x
CDC42 BPB (MRCKB )
Ser/Thr
x
CDK1/cyclin B
Ser/Thr
x
CDK2/cyclin A
Ser/Thr
x
CDK5/p25
Ser/Thr
x
CDK5/p35
Ser/Thr
x
CDK7/cyclin H/MNAT1
Ser/Thr
x
CDK8/cyclin C
Ser/Thr
x
CDK9/cyclin K
Ser/Thr
x
CDK9/cyclin T1
Ser/Thr
x
CHEK1 (CHK1 )
Ser/Thr
x
CHEK2 (CHK2 )
Ser/Thr
x
CHUK (IKK alpha )
Ser/Thr
x
CLK1
Ser/Thr
x
CLK2
Ser/Thr
x
CLK3
Ser/Thr
x
CLK4
Ser/Thr
x
CSF1R (FMS )
Tyr-R
x
CSK
Tyr-C
x
CSNK1A1 (CK1 alpha 1 )
Ser/Thr
x
CSNK1D (CK1 delta )
Ser/Thr
x
CSNK1E (CK1 epsilon )
Ser/Thr
x
CSNK1G1 (CK1 gamma 1 )
Ser/Thr
x
CSNK1G2 (CK1 gamma 2 )
Ser/Thr
x
CSNK1G3 (CK1 gamma 3 )
Ser/Thr
x
CSNK2A1 (CK2 alpha 1 )
Ser/Thr
x
CSNK2A2 (CK2 alpha 2 )
Ser/Thr
x
DAPK1
Ser/Thr
x
DAPK3 (ZIPK )
Ser/Thr
x
DCAMKL2 (DCK2 )
Ser/Thr
x
DDR1
Ser/Thr
x
DDR2
Tyr-R
x
DMPK
Ser/Thr
x
DNA-PK
Ser/Thr
x
DYRK1A
Ser/Thr
x
DYRK1B
Ser/Thr
x
DYRK3
Ser/Thr
x
DYRK4
Ser/Thr
x
EEF2K
Ser/Thr
x
EGFR (ErbB1 )
Tyr-R
x
EGFR (ErbB1) L858R
Tyr-R
x
EGFR (ErbB1) L861Q
Tyr-R
x
EGFR (ErbB1) T790M
Tyr-R
x
EGFR (ErbB1) T790M L858R
Tyr-R
x
EPHA1
Tyr-R
x
EPHA2
Tyr-R
x
EPHA3
Tyr-R
x
EPHA4
Tyr-R
x
EPHA5
Tyr-R
x
EPHA7
Tyr-R
x
EPHA8
Tyr-R
x
EPHB1
Tyr-R
x
EPHB2
Tyr-R
x
EPHB3
Tyr-R
x
EPHB4
Tyr-R
x
ERBB2 (HER2 )
Tyr-R
x
ERBB4 (HER4 )
Tyr-R
x
FER
Tyr-C
x
FES (FPS )
Tyr-C
x
FGFR1
Tyr-R
x
FGFR2
Tyr-R
x
FGFR3
Tyr-R
x
FGFR3 K650E
Tyr-R
x
FGFR4
Tyr-R
x
FGR
Tyr-C
x
FLT1 (VEGFR1 )
Tyr-R
x
FLT3
Tyr-R
x
FLT3 D835Y
Tyr-R
x
FLT4 (VEGFR3 )
Tyr-R
x
FRAP1 (mTOR )
Ser/Thr
x
FRK (PTK5 )
Tyr-C
x
FYN
Tyr-C
x
GRK4
Ser/Thr
x
GRK5
Ser/Thr
x
GRK6
Ser/Thr
x
GRK7
Ser/Thr
x
GSG2 (Haspin )
Ser/Thr
x
GSK3A (GSK3 alpha )
Ser/Thr
x
GSK3B (GSK3 beta )
Ser/Thr
x
HCK
Tyr-C
x
HIPK1 (Myak )
Ser/Thr
x
HIPK2
Ser/Thr
x
HIPK3 (YAK1 )
Ser/Thr
x
HIPK4
Ser/Thr
x
IGF1R
Tyr-R
x
IKBKB (IKK beta )
Ser/Thr
x
IKBKE (IKK epsilon )
Ser/Thr
x
INSR
Tyr-R
x
INSRR (IRR )
Tyr-R
x
IRAK1
Ser/Thr
x
IRAK4
Ser/Thr
x
ITK
Tyr-C
x
JAK1
Tyr-C
x
JAK2
Tyr-C
x
JAK2 JH1 JH2
Tyr-C
x
JAK2 JH1 JH2 V617F
Tyr-C
x
JAK3
Tyr-C
x
KDR (VEGFR2 )
Tyr-R
x
KIT
Tyr-R
x
KIT T670I
Tyr-R
x
KIT V654A
Tyr-R
x
LCK
Tyr-C
x
LIMK1
Ser/Thr
x
LIMK2
Ser/Thr
x
LRRK2
Ser/Thr
x
LRRK2 G2019S
Ser/Thr
x
LTK (TYK1 )
Tyr-R
x
LYN A
Tyr-C
x
LYN B
Tyr-C
x
MAP2K1 (MEK1 )
Ser/Thr
x
x
MAP2K1 (MEK1) S218D S222D
Ser/Thr
x
MAP2K2 (MEK2 )
Ser/Thr
x
x
MAP2K3 (MEK3 )
Ser/Thr
x
MAP2K6 (MKK6 )
Ser/Thr
x
x
MAP2K6 (MKK6) S207E T211E
Ser/Thr
x
MAP3K10 (MLK2 )
Ser/Thr
x
MAP3K11 (MLK3 )
Ser/Thr
x
MAP3K14 (NIK )
Ser/Thr
x
MAP3K2 (MEKK2 )
Ser/Thr
x
MAP3K3 (MEKK3 )
Ser/Thr
x
MAP3K5 (ASK1 )
Ser/Thr
x
MAP3K7/MAP3K7IP1 (TAK1-TAB1)
Ser/Thr
x
MAP3K8 (COT )
Ser/Thr
x
MAP3K9 (MLK1 )
Ser/Thr
x
MAP4K2 (GCK )
Ser/Thr
x
MAP4K4 (HGK )
Ser/Thr
x
MAP4K5 (KHS1 )
Ser/Thr
x
MAPK1 (ERK2 )
Ser/Thr
x
MAPK10 (JNK3 )
Ser/Thr
x
x
MAPK11 (p38 beta )
Ser/Thr
x
MAPK12 (p38 gamma )
Ser/Thr
x
MAPK13 (p38 delta )
Ser/Thr
x
MAPK14 (p38 alpha )
Ser/Thr
x
MAPK14 (p38 alpha) Direct
Ser/Thr
x
MAPK3 (ERK1 )
Ser/Thr
x
MAPK8 (JNK1 )
Ser/Thr
x
x
MAPK9 (JNK2 )
Ser/Thr
x
x
MAPKAPK2
Ser/Thr
x
MAPKAPK3
Ser/Thr
x
MAPKAPK5 (PRAK )
Ser/Thr
x
MARK1 (MARK )
Ser/Thr
x
MARK2
Ser/Thr
x
MARK3
Ser/Thr
x
MARK4
Ser/Thr
x
MATK (HYL )
Tyr-C
x
MELK
Ser/Thr
x
MERTK (cMER )
Tyr-R
x
MET (cMet )
Tyr-R
x
MET M1250T
Tyr-R
x
MINK1
Ser/Thr
x
MKNK1 (MNK1 )
Ser/Thr
x
MKNK2 (MNK2 )
Ser/Thr
x
MLCK (MLCK2 )
Ser/Thr
x
MST1R (RON )
Tyr-R
x
MST4
Ser/Thr
x
MUSK
Tyr-R
x
MYLK (MLCK )
Ser/Thr
x
MYLK2 (skMLCK )
Ser/Thr
x
NEK1
Ser/Thr
x
NEK2
Ser/Thr
x
NEK4
Ser/Thr
x
NEK6
Ser/Thr
x
NEK7
Ser/Thr
x
NEK9
Ser/Thr
x
NLK
Ser/Thr
x
NTRK1 (TRKA )
Tyr-R
x
NTRK2 (TRKB )
Tyr-R
x
NTRK3 (TRKC )
Tyr-R
x
NUAK1 (ARK5 )
Ser/Thr
x
PAK1
Ser/Thr
x
PAK2 (PAK65 )
Ser/Thr
x
PAK3
Ser/Thr
x
PAK4
Ser/Thr
x
PAK6
Ser/Thr
x
PAK7 (KIAA1264 )
Ser/Thr
x
PASK
Ser/Thr
x
PDGFRA (PDGFR alpha )
Tyr-R
x
PDGFRA D842V
Tyr-R
x
PDGFRA T674I
Tyr-R
x
PDGFRA V561D
Tyr-R
x
PDGFRB (PDGFR beta )
Tyr-R
x
PDK1
Ser/Thr
x
PDK1 Direct
Ser/Thr
x
PHKG1
Ser/Thr
x
PHKG2
Ser/Thr
x
PI4KA
Lipid
x
PI4KB (PI4K beta )
Lipid
x
PIK3C2A (PI3K-C2 alpha )
Lipid
x
PIK3C2B (PI3K-C2 beta )
Lipid
x
PIK3C3 (hVPS34 )
Lipid
x
PIK3CA/PIK3R1 (p110 alpha/p85 alpha )
Lipid
x
PIK3CD/PIK3R1 (p110 delta/p85 alpha )
Lipid
x
PIK3CG (p110 gamma )
Lipid
x
PIM1
Ser/Thr
x
PIM2
Ser/Thr
x
PKN1 (PRK1 )
Ser/Thr
x
PLK1
Ser/Thr
x
PLK2
Ser/Thr
x
PLK3
Ser/Thr
x
PRKACA (PKA )
Ser/Thr
x
PRKCA (PKC alpha )
Ser/Thr
x
PRKCB1 (PKC beta I )
Ser/Thr
x
PRKCB2 (PKC beta II )
Ser/Thr
x
PRKCD (PKC delta )
Ser/Thr
x
PRKCE (PKC epsilon )
Ser/Thr
x
PRKCG (PKC gamma )
Ser/Thr
x
PRKCH (PKC eta )
Ser/Thr
x
PRKCI (PKC iota )
Ser/Thr
x
PRKCN (PKD3 )
Ser/Thr
x
PRKCQ (PKC theta )
Ser/Thr
x
PRKCZ (PKC zeta )
Ser/Thr
x
PRKD1 (PKC mu )
Ser/Thr
x
PRKD2 (PKD2 )
Ser/Thr
x
PRKG1
Ser/Thr
x
PRKG2 (PKG2 )
Ser/Thr
x
PRKX
Ser/Thr
x
PTK2 (FAK )
Tyr-C
x
PTK2B (FAK2 )
Tyr-C
x
PTK6 (Brk )
Tyr-C
x
RAF1 (cRAF) Y340D Y341D
Ser/Thr
x
x
RET
Tyr-R
x
RET V804L
Tyr-R
x
RET Y791F
Tyr-R
x
RIPK2
Ser/Thr
x
ROCK1
Ser/Thr
x
ROCK2
Ser/Thr
x
ROS1
Tyr-R
x
RPS6KA1 (RSK1 )
Ser/Thr
x
RPS6KA2 (RSK3 )
Ser/Thr
x
RPS6KA3 (RSK2 )
Ser/Thr
x
RPS6KA4 (MSK2 )
Ser/Thr
x
RPS6KA5 (MSK1 )
Ser/Thr
x
RPS6KA6 (RSK4 )
Ser/Thr
x
RPS6KB1 (p70S6K )
Ser/Thr
x
SGK (SGK1 )
Ser/Thr
x
SGK2
Ser/Thr
x
SGKL (SGK3 )
Ser/Thr
x
SLK
Ser/Thr
x
SNF1LK2
Ser/Thr
x
SPHK1
Lipid
x
SPHK2
Lipid
x
SRC
Tyr-C
x
SRC N1
Tyr-C
x
SRMS (Srm )
Tyr-C
x
SRPK1
Ser/Thr
x
SRPK2
Ser/Thr
x
STK16 (PKL12 )
Ser/Thr
x
STK17A (DRAK1 )
Ser/Thr
x
STK22B (TSSK2 )
Ser/Thr
x
STK22D (TSSK1 )
Ser/Thr
x
STK23 (MSSK1 )
Ser/Thr
x
STK24 (MST3 )
Ser/Thr
x
STK25 (YSK1 )
Ser/Thr
x
STK3 (MST2 )
Ser/Thr
x
STK33
Ser/Thr
x
STK4 (MST1 )
Ser/Thr
x
SYK
Tyr-C
x
TAOK2 (TAO1 )
Ser/Thr
x
TAOK3 (JIK )
Ser/Thr
x
TBK1
Ser/Thr
x
TEC
Tyr-C
x
TEK (Tie2 )
Tyr-R
x
TGFBR1 (ALK5 )
Ser/Thr
x
TNK2 (ACK )
Tyr-C
x
TTK
Ser/Thr
x
TXK
Tyr-C
x
TYK2
Tyr-C
x
TYRO3 (RSE )
Tyr-R
x
WEE1
Ser/Thr
x
WNK2
Ser/Thr
x
YES1
Tyr-C
x
ZAK
Ser/Thr
x
ZAP70
Tyr-C
x