Kinase
Activity Assays
Binding Assay
Z'-LYTE®
Adapta®
LanthaScreen®
AXL
x
CSF1R (FMS )
x
DDR2
x
EGFR (ErbB1 )
x
EGFR (ErbB1) L858R
x
EGFR (ErbB1) L861Q
x
EGFR (ErbB1) T790M
x
EGFR (ErbB1) T790M L858R
x
EPHA1
x
EPHA2
x
EPHA3
x
EPHA4
x
EPHA5
x
EPHA7
x
EPHA8
x
EPHB1
x
EPHB2
x
EPHB3
x
EPHB4
x
ERBB2 (HER2 )
x
ERBB4 (HER4 )
x
FGFR1
x
FGFR2
x
FGFR3
x
FGFR3 K650E
x
FGFR4
x
FLT1 (VEGFR1 )
x
FLT3
x
FLT3 D835Y
x
FLT4 (VEGFR3 )
x
IGF1R
x
INSR
x
INSRR (IRR )
x
KDR (VEGFR2 )
x
KIT
x
KIT T670I
x
KIT V654A
x
LTK (TYK1 )
x
MERTK (cMER )
x
MET (cMet )
x
MET M1250T
x
MST1R (RON )
x
MUSK
x
NTRK1 (TRKA )
x
NTRK2 (TRKB )
x
NTRK3 (TRKC )
x
PDGFRA (PDGFR alpha )
x
PDGFRA D842V
x
PDGFRA T674I
x
PDGFRA V561D
x
PDGFRB (PDGFR beta )
x
RET
x
RET V804L
x
RET Y791F
x
ROS1
x
TEK (Tie2 )
x
TYRO3 (RSE )
x