Target Name

Cell Background

Stimulus

Androgen Receptor (AR)

GripTite™ 293

R1881

Estrogen Receptor-alpha (ER-alpha)

GripTite™ 293

17-beta-Estradiol

Estrogen Receptor-beta (ER-beta)

GripTite™ 293

17-beta-Estradiol

Estrogen Related Receptor-alpha (ERR-alpha)

HEK 293T

None

Farnesoid X Receptor (FXR)

HEK 293T

Chenodeoxycholic Acid

Glucocorticoid Receptor (GR)

HEK 293T

Dexamethasone

Liver X Receptor Alpha (LXR-alpha)

HEK 293T

TO901317

Liver X Receptor Beta (LXR-beta)

HEK 293T

TO901317

Mineralcorticoid Receptor (MR)

HEK 293T

Aldosterone

Peroxisome Proliferator Activated Receptor Delta (PPAR-delta)

HEK 293T

L-165041

Peroxisome Proliferator Activated Receptor-gamma (PPAR-gamma)

HEK 293H

Rosiglitazone

Progesterone Receptor (PR)

HEK 293T

R5020

Retinoic Acid Receptor Alpha (RAR-alpha)

HEK 293T

ATRA

Retinoic Acid Receptor Beta (RAR-beta)

HEK 293T

ATRA

Retinoic Acid Receptor Gamma (RAR-gamma)

HEK 293T

ATRA

Retinoid X Receptor-alpha (RXR-alpha)

HEK 293T

9-cis retinoic acid

Retinoid X Receptor-beta (RXR-beta)

HEK 293T

9-cis retinoic acid

Thyroid Hormone Receptor-alpha (TR-alpha)

HEK 293T

T3 Sodium Salt

Thyroid Hormone Receptor-beta (TR-beta)

HEK 293T

T3 Free Acid

Vitamin D Receptor (VDR)

HEK 293T

Calcitriol